BindingDB BDBM4552 4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methyl-1-piperazinyl)propoxy]-3-quinolinecarbonitrile::4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile::BOSUTINIB::CHEMBL288441::SKI-606

BDBM4552 4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methyl-1-piperazinyl)propoxy]-3-quinolinecarbonitrile::4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile::BOSUTINIB::CHEMBL288441::SKI-606

SMILES COc1cc(Nc2c(cnc3cc(OCCCN4CCN(C)CC4)c(OC)cc23)C#N)c(Cl)cc1Cl

InChI Key InChIKey=UBPYILGKFZZVDX-UHFFFAOYSA-N

Data 5 KI 93 IC50 456 Kd

PDB links: 14 PDB IDs match this monomer.

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 4552

Protein kinase C eta type(Homo sapiens (Human))
Ambit Biosciences

Curated by ChEMBL

BDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)

Kd: >1.00E+4nMAssay Description:Binding constant for PRKCH kinase domainMore data for this Ligand-Target Pair

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Targets 382▿
- Proto-oncogene tyrosine-protein kinase Src 29
- Tyrosine-protein kinase ABL1 21
- Epidermal growth factor receptor 14
- Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase 11
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform 10
- Mast/stem cell growth factor receptor Kit 9
- Receptor-type tyrosine-protein kinase FLT3 7
- Tyrosine-protein kinase receptor UFO 5
- Proto-oncogene tyrosine-protein kinase receptor Ret 4
- Activated CDC42 kinase 1 4
- ALK tyrosine kinase receptor/Nucleophosmin 4
- Cytoplasmic tyrosine-protein kinase BMX 3
- Wee1-like protein kinase 3
- Cyclin-G-associated kinase 3
- Serine/threonine-protein kinase TBK1 3
- Hepatocyte growth factor receptor 3
- Tyrosine-protein kinase Fyn 3
- Tyrosine-protein kinase Lyn 3
- Tyrosine-protein kinase Fer 2
- Tyrosine-protein kinase Tec 2
- Tyrosine-protein kinase JAK1 2
- Cyclin-dependent kinase 4 2
- Tyrosine-protein kinase FRK 2
- Angiopoietin-1 receptor 2
- Mitogen-activated protein kinase kinase kinase kinase 2 2
- Mitogen-activated protein kinase kinase kinase kinase 3 2
- Mitogen-activated protein kinase kinase kinase kinase 5 2
- Non-receptor tyrosine-protein kinase TYK2 2
- Mitogen-activated protein kinase 14 2
- Serine/threonine-protein kinase B-raf 2
- Interleukin-1 receptor-associated kinase 4 2
- Tyrosine-protein kinase ABL2 2
- Dual specificity mitogen-activated protein kinase kinase 1 2
- Serine/threonine-protein kinase 10 2
- Breakpoint cluster region protein/Tyrosine-protein kinase ABL1 2
- Leucine-rich repeat serine/threonine-protein kinase 2 2
- Tyrosine-protein kinase Fes/Fps 2
- BDNF/NT-3 growth factors receptor 2
- Tyrosine-protein kinase Lck 2
- Serine/threonine-protein kinase 4 2
- Tyrosine-protein kinase BTK 2
- Dual specificity protein kinase CLK1 2
- Ephrin type-A receptor 2 [596-900] 2
- Ephrin type-A receptor 6 2
- Dual specificity protein kinase CLK3 2
- Dual specificity protein kinase CLK2 2
- High affinity nerve growth factor receptor 2
- Protein-tyrosine kinase 2-beta 2
- Tyrosine-protein kinase Blk 2
- Calcium/calmodulin-dependent protein kinase type II subunit gamma 2
- Tyrosine-protein kinase SYK 2
- Ribosomal protein S6 kinase alpha-2 2
- Ribosomal protein S6 kinase alpha-1 2
- Calcium/calmodulin-dependent protein kinase type 1D 2
- Tyrosine-protein kinase Fgr 2
- Tyrosine-protein kinase HCK 2
- Fibroblast growth factor receptor 3 2
- Wee1-like protein kinase 2 2
- Misshapen-like kinase 1 2
- Tyrosine-protein kinase CSK 2
- Ribosomal protein S6 kinase alpha-6 2
- Focal adhesion kinase 1 2
- Serine/threonine-protein kinase 24 2
- Ribosomal protein S6 kinase alpha-4 2
- Ribosomal protein S6 kinase alpha-5 2
- Ephrin type-B receptor 4 2
- Ephrin type-B receptor 2 2
- Tyrosine-protein kinase TXK 2
- Tyrosine-protein kinase Yes 2
- BMP-2-inducible protein kinase 1
- Rhodopsin kinase GRK1 1
- Cyclin-dependent kinase 11B 1
- Cyclin-dependent kinase 11A 1
- Uncharacterized serine/threonine-protein kinase SBK3 1
- LIM domain kinase 1 1
- LIM domain kinase 2 1
- ALK tyrosine kinase receptor 1
- NUAK family SNF1-like kinase 2 1
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform 1
- Glycogen synthase kinase-3 beta 1
- Calcium/calmodulin-dependent protein kinase type 1 1
- Protein kinase C iota type 1
- NUAK family SNF1-like kinase 1 1
- Transient receptor potential cation channel subfamily M member 6 1
- AP2-associated protein kinase 1 1
- Calcium/calmodulin-dependent protein kinase type II subunit beta 1
- Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform 1
- Serine/threonine-protein kinase PAK 1 1
- Protein kinase C theta type 1
- Serine/threonine-protein kinase PAK 2 1
- Serine/threonine-protein kinase PAK 3 1
- Dual specificity mitogen-activated protein kinase kinase 2 1
- Serine/threonine-protein kinase PAK 4 1
- Phosphatidylinositol 5-phosphate 4-kinase type-2 beta 1
- Serine/threonine-protein kinase tousled-like 2 1
- Dual specificity mitogen-activated protein kinase kinase 3 1
- Serine/threonine-protein kinase PAK 5 1
- Serine/threonine-protein kinase PAK 6 1
- Serine/threonine-protein kinase tousled-like 1 1
- Tyrosine-protein kinase JAK3 1
- Tyrosine-protein kinase JAK2 1
- Dual specificity mitogen-activated protein kinase kinase 6 1
- Dual specificity mitogen-activated protein kinase kinase 7 1
- Dual specificity mitogen-activated protein kinase kinase 4 1
- Dual specificity mitogen-activated protein kinase kinase 5 1
- Tyrosine-protein kinase ZAP-70 1
- Casein kinase I isoform gamma-3 1
- Casein kinase I isoform gamma-2 1
- Serine/threonine-protein kinase Sgk3 1
- Casein kinase I isoform epsilon 1
- Casein kinase I isoform gamma-1 1
- Myosin light chain kinase 3 1
- Ephrin type-A receptor 1 1
- Ephrin type-A receptor 3 1
- Ephrin type-A receptor 2 1
- Ephrin type-A receptor 5 1
- Ephrin type-A receptor 4 1
- Insulin-like growth factor 1 receptor 1
- Activin receptor type-1 1
- Myosin light chain kinase 2, skeletal/cardiac muscle 1
- Tyrosine-protein kinase Srms 1
- Serine/threonine-protein kinase/endoribonuclease IRE1 1
- Serine/threonine-protein kinase MAK 1
- Phosphatidylinositol 3-kinase C2 domain-containing subunit gamma 1
- Ankyrin repeat and protein kinase domain-containing protein 1 1
- Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma 1
- Cyclin-dependent kinase 2 1
- Rhodopsin kinase GRK7 1
- Ephrin type-A receptor 8 1
- Phosphatidylinositol 4-kinase beta 1
- Death-associated protein kinase 2 1
- Death-associated protein kinase 1 1
- Serine/threonine-protein kinase D2 1
- Serine/threonine-protein kinase D3 1
- TGF-beta receptor type-2 1
- Serine/threonine-protein kinase D1 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 1B 1
- Dual serine/threonine and tyrosine protein kinase 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 1A 1
- Death-associated protein kinase 3 1
- Cyclin-dependent kinase 9 1
- Serine/threonine-protein kinase pim-3 1
- Cyclin-dependent kinase 8 1
- Cyclin-dependent kinase 7 1
- Serine/threonine-protein kinase pim-1 1
- Cyclin-dependent kinase 5 1
- Serine/threonine-protein kinase pim-2 1
- Serine/threonine-protein kinase 38 1
- Serine/threonine-protein kinase 35 1
- Cyclin-dependent kinase 3 1
- Serine/threonine-protein kinase 36 1
- Cyclin-dependent kinase 16 1
- Testis-specific serine/threonine-protein kinase 1 1
- Protein kinase C epsilon type 1
- Cyclin-dependent kinase 17 1
- Bone morphogenetic protein receptor type-2 1
- Cyclin-dependent kinase 19 1
- Cyclin-dependent kinase 2 homolog 1
- Protein-tyrosine kinase 6 1
- Casein kinase II subunit alpha 1
- Cyclin-dependent kinase 13 1
- Cyclin-dependent kinase 14 1
- Cyclin-dependent kinase 15 1
- Leukocyte tyrosine kinase receptor 1
- Atypical kinase COQ8B, mitochondrial 1
- Tyrosine-protein kinase ABL1/ABL2 1
- Microtubule-associated serine/threonine-protein kinase 1 1
- Calcium/calmodulin-dependent protein kinase type II subunit alpha 1
- cGMP-dependent protein kinase 2 1
- Rho-associated protein kinase 2 1
- cGMP-dependent protein kinase 1 1
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform 1
- Rho-associated protein kinase 1 1
- Serine/threonine-protein kinase ULK1 1
- Serine/threonine-protein kinase SIK2 1
- Serine/threonine-protein kinase SIK1 1
- Serine/threonine-protein kinase ULK2 1
- Serine/threonine-protein kinase ULK3 1
- 3-phosphoinositide-dependent protein kinase 1 1
- Mitogen-activated protein kinase 1 1
- Serine/threonine-protein kinase 3 1
- Mitogen-activated protein kinase 3 1
- Discoidin domain-containing receptor 2 1
- Mitogen-activated protein kinase 4 1
- SRSF protein kinase 3 1
- Mitogen-activated protein kinase 9 1
- SRSF protein kinase 2 1
- Mitogen-activated protein kinase 6 1
- Mitogen-activated protein kinase 7 1
- Calcium/calmodulin-dependent protein kinase type IV 1
- Mitogen-activated protein kinase 8 1
- Serine/threonine-protein kinase RIO1 1
- Serine/threonine-protein kinase LATS1 1
- Serine/threonine-protein kinase RIO3 1
- Serine/threonine-protein kinase 32B 1
- Serine/threonine-protein kinase RIO2 1
- Serine/threonine-protein kinase 32A 1
- Serine/threonine-protein kinase 32C 1
- Vascular endothelial growth factor receptor 2 1
- Insulin receptor 1
- Vascular endothelial growth factor receptor 3 1
- Vascular endothelial growth factor receptor 1 1
- Serine/threonine-protein kinase PLK1 1
- Serine/threonine-protein kinase PLK2 1
- Insulin receptor-related protein 1
- Inhibitor of nuclear factor kappa-B kinase subunit beta 1
- Serine/threonine-protein kinase NIM1 1
- Serine/threonine-protein kinase PLK3 1
- Serine/threonine-protein kinase PLK4 1
- Tyrosine-protein kinase receptor TYRO3 1
- Serine/threonine-protein kinase BRSK1 1
- Serine/threonine-protein kinase LATS2 1
- cAMP-dependent protein kinase catalytic subunit alpha 1
- Citron Rho-interacting kinase 1
- Platelet-derived growth factor receptor alpha 1
- Serine/threonine-protein kinase BRSK2 1
- Serine/threonine-protein kinase Chk2 1
- Serine/threonine-protein kinase Chk1 1
- cAMP-dependent protein kinase catalytic subunit PRKX 1
- SRSF protein kinase 1 1
- Serine/threonine-protein kinase MRCK beta 1
- Serine/threonine-protein kinase MRCK gamma 1
- Casein kinase II subunit alpha' 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 2 1
- Serine/threonine-protein kinase STK11 1
- Peripheral plasma membrane protein CASK 1
- Receptor tyrosine-protein kinase erbB-4 1
- Receptor tyrosine-protein kinase erbB-2 1
- Receptor tyrosine-protein kinase erbB-3 1
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform 1
- Serine/threonine-protein kinase Nek9 1
- Serine/threonine-protein kinase Nek7 1
- Glycogen synthase kinase-3 alpha 1
- Serine/threonine-protein kinase Nek6 1
- Serine/threonine-protein kinase Nek5 1
- Serine/threonine-protein kinase Nek4 1
- Serine/threonine-protein kinase Nek3 1
- Serine/threonine-protein kinase Nek2 1
- Serine/threonine-protein kinase receptor R3 1
- Serine/threonine-protein kinase Nek1 1
- Macrophage-stimulating protein receptor 1
- Cyclin-dependent kinase-like 3 1
- Serine/threonine-protein kinase SIK3 [59-1321] 1
- Cyclin-dependent kinase-like 2 1
- MAP/microtubule affinity-regulating kinase 3 1
- Homeodomain-interacting protein kinase 4 1
- Homeodomain-interacting protein kinase 3 1
- MAP kinase-interacting serine/threonine-protein kinase 2 1
- MAP kinase-interacting serine/threonine-protein kinase 1 1
- Cyclin-dependent kinase-like 5 1
- MAP/microtubule affinity-regulating kinase 4 1
- Serine/threonine-protein kinase 38-like 1
- Dual specificity protein kinase TTK 1
- Myosin-IIIb 1
- Serine/threonine-protein kinase Nek11 1
- Myosin-IIIa 1
- Eukaryotic translation initiation factor 2-alpha kinase 1 1
- Serine/threonine-protein kinase mTOR 1
- Tyrosine-protein kinase ITK/TSK 1
- Myotonin-protein kinase 1
- Protein kinase C eta type 1
- Bone morphogenetic protein receptor type-1B 1
- Bone morphogenetic protein receptor type-1A 1
- Receptor-interacting serine/threonine-protein kinase 1 1
- Serine/threonine-protein kinase 16 1
- Receptor-interacting serine/threonine-protein kinase 2 1
- SNF-related serine/threonine-protein kinase 1
- Non-receptor tyrosine-protein kinase TNK1 1
- Inhibitor of nuclear factor kappa-B kinase subunit epsilon 1
- Serine/threonine-protein kinase NLK 1
- Homeodomain-interacting protein kinase 2 1
- Homeodomain-interacting protein kinase 1 1
- Receptor-interacting serine/threonine-protein kinase 4 1
- Ribosomal protein S6 kinase beta-1 1
- Serine/threonine-protein kinase OSR1 1
- Casein kinase I isoform delta 1
- Cyclin-dependent kinase 18 [3-474] 1
- RAF proto-oncogene serine/threonine-protein kinase 1
- Serine/threonine-protein kinase 26 1
- Serine/threonine-protein kinase 25 1
- Dual specificity testis-specific protein kinase 1 1
- Ephrin type-B receptor 3 1
- Serine/threonine-protein kinase 33 1
- Ephrin type-B receptor 1 1
- Serine/threonine-protein kinase SBK1 1
- MAP kinase-activated protein kinase 2 1
- Ephrin type-B receptor 6 1
- Platelet-derived growth factor receptor beta 1
- Epithelial discoidin domain-containing receptor 1 1
- MAP kinase-activated protein kinase 5 1
- STE20/SPS1-related proline-alanine-rich protein kinase 1
- Muscle, skeletal receptor tyrosine-protein kinase 1
- Calcium-dependent protein kinase 1 1
- Tyrosine-protein kinase receptor Tie-1 1
- 5'-AMP-activated protein kinase catalytic subunit alpha-2 1
- Calcium/calmodulin-dependent protein kinase type II subunit delta 1
- Proto-oncogene tyrosine-protein kinase ROS 1
- Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma 1
- Serine/threonine-protein kinase TAO1 1
- Serine/threonine-protein kinase DCLK1 1
- Calcium/calmodulin-dependent protein kinase kinase 1 1
- Serine/threonine-protein kinase PknB 1
- Serine/threonine-protein kinase DCLK2 1
- Serine/threonine-protein kinase TAO3 1
- Serine/threonine-protein kinase PRP4 homolog 1
- Calcium/calmodulin-dependent protein kinase kinase 2 1
- Serine/threonine-protein kinase TAO2 1
- Serine/threonine-protein kinase DCLK3 1
- Serine/threonine-protein kinase TNNI3K 1
- Interferon-induced, double-stranded RNA-activated protein kinase 1
- Cyclin-dependent kinase-like 1 [2-358] 1
- Mitogen-activated protein kinase kinase kinase kinase 1 1
- Serine/threonine-protein kinase MRCK alpha 1
- Casein kinase I isoform alpha-like 1
- Mitogen-activated protein kinase kinase kinase kinase 4 1
- Mitogen-activated protein kinase 15 1
- Broad substrate specificity ATP-binding cassette transporter ABCG2 1
- 5'-AMP-activated protein kinase catalytic subunit alpha-1 1
- Activin receptor type-1B 1
- Myosin light chain kinase family member 4 1
- Mitogen-activated protein kinase kinase kinase 9 1
- Serine/threonine-protein kinase VRK2 1
- Mitogen-activated protein kinase kinase kinase 6 1
- RAC-gamma serine/threonine-protein kinase 1
- Mitogen-activated protein kinase kinase kinase 5 1
- Interleukin-1 receptor-associated kinase 1 1
- Mitogen-activated protein kinase kinase kinase 7 1
- Interleukin-1 receptor-associated kinase 3 1
- Mitogen-activated protein kinase kinase kinase 2 1
- Mitogen-activated protein kinase kinase kinase 1 1
- Mitogen-activated protein kinase kinase kinase 4 1
- Mitogen-activated protein kinase kinase kinase 3 1
- Serine/threonine-protein kinase ICK 1
- RAC-alpha serine/threonine-protein kinase 1
- Megakaryocyte-associated tyrosine-protein kinase 1
- Activin receptor type-2B 1
- Myosin light chain kinase, smooth muscle 1
- Activin receptor type-2A 1
- Serine/threonine-protein kinase 17A 1
- Serine/threonine-protein kinase 17B 1
- Mitogen-activated protein kinase kinase kinase 19 1
- Protein kinase C delta type 1
- Mitogen-activated protein kinase kinase kinase 15 1
- NT-3 growth factor receptor 1
- G protein-coupled receptor kinase 4 1
- Dual specificity protein kinase CLK4 1
- Tyrosine-protein kinase Mer 1
- Serine/threonine-protein kinase N2 1
- cAMP-dependent protein kinase catalytic subunit beta 1
- Serine/threonine-protein kinase N1 1
- Ribosomal protein S6 kinase alpha-3 1
- Phosphorylase b kinase gamma catalytic chain, liver/testis isoform 1
- STE20-like serine/threonine-protein kinase 1
- Calcium/calmodulin-dependent protein kinase type 1G 1
- Hormonally up-regulated neu tumor-associated kinase 1
- Fibroblast growth factor receptor 4 1
- Aurora kinase B 1
- Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta 1
- Aurora kinase A 1
- Mitogen-activated protein kinase kinase kinase 20 1
- Fibroblast growth factor receptor 1 1
- Fibroblast growth factor receptor 2 1
- Atypical kinase COQ8A, mitochondrial 1
- Aurora kinase C 1
- Mitogen-activated protein kinase 13 1
- Inhibitor of nuclear factor kappa-B kinase subunit alpha 1
- Mitogen-activated protein kinase 12 1
- Mitogen-activated protein kinase 11 1
- Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha 1
- RAC-beta serine/threonine-protein kinase 1
- Mitogen-activated protein kinase 10 1
- Casein kinase I isoform alpha 1
- Macrophage colony-stimulating factor 1 receptor 1
- eIF-2-alpha kinase GCN2 1
- Maternal embryonic leucine zipper kinase 1
- Serine/threonine-protein kinase MARK1 1
- Serine/threonine-protein kinase MARK2 1
- TRAF2 and NCK-interacting protein kinase 1
- Mitogen-activated protein kinase kinase kinase 12 1
- Mitogen-activated protein kinase kinase kinase 13 1
- Mitogen-activated protein kinase kinase kinase 10 1
- Mitogen-activated protein kinase kinase kinase 11 1
- ...
Publications 37▿
- Nat Biotechnol 29: 1046-51 (2011) 442
- Leukemia 23: 477-85 (2009) 41
- J Med Chem 59: 3593-608 (2016) 6
- Eur J Med Chem 161: 479-492 (2019) 5
- J Med Chem 49: 5759-68 (2006) 5
- Bioorg Med Chem 26: 4014-4024 (2018) 4
- Bioorg Med Chem Lett 13: 2977-80 (2003) 3
- Eur J Med Chem 126: 754-761 (2017) 3
- J Med Chem 60: 7863-7875 (2017) 3
- J Med Chem 62: 4772-4778 (2019) 2
- ACS Chem Biol 11: 3400-3411 (2016) 2
- Bioorg Med Chem Lett 29: 1727-1731 (2019) 2
- J Med Chem 48: 3891-902 (2005) 2
- Bioorg Med Chem Lett 18: 6206-9 (2008) 2
- J Med Chem 53: 1413-37 (2010) 2
- Eur J Med Chem 238: (2022) 2
- Bioorg Med Chem Lett 20: 2924-7 (2010) 2
- J Med Chem 48: 6523-43 (2005) 2
- Bioorg Med Chem Lett 19: 5071-4 (2009) 2
- J Med Chem 65: 893-921 (2022) 2
- J Med Chem 47: 1599-601 (2004) 2
- J Med Chem 58: 2746-63 (2015) 1
- Bioorg Med Chem 19: 2517-28 (2011) 1
- Bioorg Med Chem 16: 5890-8 (2008) 1
- Eur J Med Chem 237: (2022) 1
- J Med Chem 61: 6277-6292 (2018) 1
- J Med Chem 65: 935-954 (2022) 1
- J Med Chem 49: 7868-76 (2006) 1
- J Med Chem 59: 1984-2004 (2016) 1
- Bioorg Med Chem Lett 12: 2011-4 (2002) 1
- Bioorg Med Chem 17: 3152-61 (2009) 1
- J Med Chem 47: 6666-8 (2004) 1
- J Med Chem 48: 5909-20 (2005) 1
- J Med Chem 44: 3965-77 (2001) 1
- Bioorg Med Chem Lett 15: 1743-7 (2005) 1
- Bioorg Med Chem Lett 28: 1964-1971 (2018) 1
- ACS Chem Biol 10: 289-98 (2015) 1
Institutions 25▿
- Ambit Biosciences 442
- Center For Molecular Medicine Of The Austrian Academy Of Sciences 41
- Wyeth Research 15
- Martin-Luther-University Halle-Wittenberg 9
- University Of Edinburgh 6
- University Of Milano-Bicocca 5
- University Of North Carolina At Chapel Hill 4
- China Pharmaceutical University 3
- Moffitt Cancer Center 3
- Comenius University In Bratislava 3
- Schering-Plough 2
- Csir-Indian Institute Of Integrative Medicine 2
- Organon Laboratories 2
- Technical University of Munich 2
- Wyeth-Ayerst Research 2
- Hangzhou Medical College 2
- Centro De Investigaciones Biol�Gicas Margarita Salas (Csic) 1
- Biogen 1
- High Magnetic Field Laboratory 1
- Konkuk University 1
- Vichem Chemie Research 1
- Institut De Recherches Servier 1
- Technical University of Dortmund 1
- Federal University Of Parana 1
- University Of South Florida 1
Affinity: 0.029 to 2.0E+4 nM▿
- Ki 5
- IC50 93
- Kd 456
- Affinity ≤ nM
Xtal structures: 1
Docked structures: 0
Catalog Cmpds: 1